Publications by the researcher in collaboration with FRANCISCO JAVIER SARDINA LOPEZ (9)

2021

  1. 3,4-Dihydropyrimidin-2(1H)-ones as Antagonists of the Human A2B Adenosine Receptor: Optimization, Structure-Activity Relationship Studies, and Enantiospecific Recognition

    Journal of medicinal chemistry, Vol. 64, Núm. 1, pp. 458-480

2008

  1. Design, synthesis, evaluation, and crystallographic-based structural studies of HIV-1 protease inhibitors with reduced response to the V82A mutation

    Journal of Medicinal Chemistry, Vol. 51, Núm. 4, pp. 852-860

2000

  1. A short, efficient, and stereoselective procedure for the synthesis of cis-3-hydroxymethyl-aziridine-2-carboxylic acid derivatives, important intermediates in the synthesis of mitomycinoids

    Journal of Organic Chemistry, Vol. 65, Núm. 20, pp. 6780-6783

1997

  1. Enantiomerically Pure Highly Functionalized α-Amino Ketones from the Reaction of Chiral Cyclic N-(9-Phenylfluoren-9-yl) α-Amido Esters with Organolithium Reagents

    Journal of Organic Chemistry, Vol. 62, Núm. 14, pp. 4770-4779

  2. Enantiospecific synthesis of γ-keto-α,β-diamino acid derivatives. Stereoselective synthesis of a precursor of streptolidine lactam

    Tetrahedron Letters, Vol. 38, Núm. 4, pp. 673-676

1996

  1. A versatile, enantioselective, stereocontrolled synthesis of (1S,2R)-imidazoleglycerol

    Tetrahedron Letters, Vol. 37, Núm. 51, pp. 9259-9262

1994

  1. On the Stereoselectivity of the Reaction of N-(9-Phenylfluoren-9-yl)aspartate Enolates with Electrophiles. Synthesis of Enantiomerically Pure 3-Hydroxy-, 3-Amino-, and 3-Hydroxy-3-methylaspartates

    Journal of Organic Chemistry, Vol. 59, Núm. 25, pp. 7643-7652

1992

  1. A stereodivergent chirospecific synthesis of (3R) and (3S) 3-hydroxyaspartates by hydroxylation of aspartate diester enolates

    Tetrahedron Letters, Vol. 33, Núm. 32, pp. 4637-4640

1986

  1. Complete Structural Analysis of Cyclic Polyhalogenated Monoterpenes. A Force Field 2D NMR Study

    Journal of Organic Chemistry, Vol. 51, Núm. 25, pp. 4970-4973