Instituto de Materiais (iMATUS)
Instituto
José Manuel
Brea Floriani
Profesor titular de universidade
Publicacións nas que colabora con José Manuel Brea Floriani (13)
2023
-
Design and biopharmaceutical preclinical characterisation of a new thermosensitive hydrogel for the removal of gastric polyps
International Journal of Pharmaceutics, Vol. 635, pp. 122706
-
Exploring the Effect of Halogenation in a Series of Potent and Selective A2BAdenosine Receptor Antagonists
Journal of Medicinal Chemistry, Vol. 66, Núm. 1, pp. 890-912
2017
-
3-Oxopyridazin-5-yl-Chalcone Hybrids: Potent Antiplatelet Agents That Prevent Glycoprotein IIb/IIIa Activation
ChemistrySelect, Vol. 2, Núm. 17, pp. 4920-4933
2013
-
Cytocompatibility and P-glycoprotein inhibition of block copolymers: Structure-activity relationship
Molecular Pharmaceutics, Vol. 10, Núm. 8, pp. 3232-3241
-
Discovery of 3,4-dihydropyrimidin-2(1 H)-ones as a novel class of potent and selective A2B adenosine receptor antagonists
ACS Medicinal Chemistry Letters, Vol. 4, Núm. 11, pp. 1031-1036
-
Doxorubicin-loaded micelles of reverse poly(butylene oxide)-poly(ethylene oxide)-poly(butylene oxide) block copolymers as efficient "active" chemotherapeutic agents
International Journal of Pharmaceutics, Vol. 445, Núm. 1-2, pp. 47-57
-
Poly(styrene oxide)-poly(ethylene oxide) block copolymers: From "classical" chemotherapeutic nanocarriers to active cell-response inducers
Journal of Controlled Release, Vol. 167, Núm. 1, pp. 68-75
-
Selective and potent adenosine A3 receptor antagonists by methoxyaryl substitution on the N-(2,6-diarylpyrimidin-4-yl)acetamide scaffold
European Journal of Medicinal Chemistry, Vol. 59, pp. 235-242
2012
-
Polyethylene oxide-polystyrene oxide triblock copolymers as biological-responsive nanocarriers
Materials Research Society Symposium Proceedings
2011
-
Pyrimidine derivatives as potent and selective A3 adenosine receptor antagonists
Journal of Medicinal Chemistry, Vol. 54, Núm. 2, pp. 457-471
2010
-
Inhibition of P-glycoprotein pumps by PEO-PPO amphiphiles: Branched versus linear derivatives
Nanomedicine, Vol. 5, Núm. 9, pp. 1371-1383
2009
-
Divergent solution-phase synthesis of diarylpyrimidine libraries as selective A3 adenosine receptor antagonists
Journal of Combinatorial Chemistry, Vol. 11, Núm. 4, pp. 519-522
2005
-
Synthesis and binding affinity of novel 3-aminoethyl-1-tetralones, potential atypical antipsychotics
Bioorganic and Medicinal Chemistry Letters, Vol. 15, Núm. 12, pp. 3063-3066