Instituto de Materiais (iMATUS)
Instituto
ROMAN
PEREZ FERNANDEZ
Catedrático de universidade
Publicacións nas que colabora con ROMAN PEREZ FERNANDEZ (14)
2024
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First Sila-Vitamin D Analogues: Design, Synthesis, Structural Analysis and Biological Activity
Journal of Medicinal Chemistry, Vol. 67, Núm. 23, pp. 21505-21519
2023
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Further Studies on the Highly Active Des-C-Ring and Aromatic-D-Ring Analogues of 1α,25-Dihydroxyvitamin D3 (Calcitriol): Refinement of the Side Chain
Journal of Medicinal Chemistry, Vol. 66, Núm. 22, pp. 15326-15339
2022
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Design, Synthesis, Biological Activity, and Structural Analysis of Novel Des-C-Ring and Aromatic-D-Ring Analogues of 1α,25-Dihydroxyvitamin D3
Journal of Medicinal Chemistry, Vol. 65, Núm. 19, pp. 13112-13124
2021
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Anti-inflammatory effect of tacrolimus/hydroxypropyl-β-cyclodextrin eye drops in an endotoxin-induced uveitis model
Pharmaceutics, Vol. 13, Núm. 10
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Tailored hydrogels as delivery platforms for conditioned medium from mesenchymal stem cells in a model of acute colitis in mice
Pharmaceutics, Vol. 13, Núm. 8
2019
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Mesenchymal stem cells in homeostasis and systemic diseases: Hypothesis, evidences, and therapeutic opportunities
International Journal of Molecular Sciences, Vol. 20, Núm. 15
2018
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Aromatic-Based Design of Highly Active and Noncalcemic Vitamin D Receptor Agonists
Journal of Medicinal Chemistry, Vol. 61, Núm. 11, pp. 4928-4937
2016
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Carborane-based design of a potent Vitamin D receptor agonist
Chemical Science, Vol. 7, Núm. 2, pp. 1033-1037
2015
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Pit-1 inhibits BRCA1 and sensitizes human breast tumors to cisplatin and vitamin D treatment
Oncotarget, Vol. 6, Núm. 16, pp. 14456-14471
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Synthesis and biological activity of two C.7 methyl analogues of Vitamin D
Journal of Organic Chemistry, Vol. 80, Núm. 1, pp. 165-173
2014
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26,26,26,27,27,27-hexadeuterated-1,25-dihydroxyvitamin D3 (1,25D-d6) as adjuvant of chemotherapy in breast cancer cell lines
Cancers, Vol. 6, Núm. 1, pp. 67-78
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Synthesis of nonadeuterated 1α,25-dihydroxyvitamin D2
Journal of Steroid Biochemistry and Molecular Biology, Vol. 144, Núm. PART A, pp. 204-206
2013
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Administration of the optimized β-Lapachone-poloxamer-cyclodextrin ternary system induces apoptosis, DNA damage and reduces tumor growth in a human breast adenocarcinoma xenograft mouse model
European Journal of Pharmaceutics and Biopharmaceutics, Vol. 84, Núm. 3, pp. 497-504
2012
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Synthesis and biological evaluation of 1α,25-dihydroxyvitamin D 3 analogues with a long side chain at C12 and short C17 side chains
Journal of Medicinal Chemistry, Vol. 55, Núm. 20, pp. 8642-8656