JORGE CHRISTIAN
FERNANDEZ MASAGUER
Profesor titular de universidade
JOSE ANGEL
FONTENLA GIL
Profesor titular de universidade
Publikationen, an denen er mitarbeitet JOSE ANGEL FONTENLA GIL (7)
2000
-
Butyrophenone analogues in the carbazole series as potential atypical antipsychotics: Synthesis and determination of affinities at D2, 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors
European Journal of Medicinal Chemistry, Vol. 35, Núm. 1, pp. 83-95
-
Conformationally constrained butyrophenones with affinity for dopamine (D1, D2, D4) and serotonin (5-HT(2A), 5-HT(2B), 5-HT(2C)) receptors: Synthesis of aminomethylbenzo[b]furanones and their evaluation as antipsychotics
Journal of Medicinal Chemistry, Vol. 43, Núm. 24, pp. 4678-4693
1999
-
Conformationally constrained butyrophenones with mixed dopaminergic (D2) and serotoninergic (5-HT2(A), 5-HT2(C)) affinities: Synthesis, pharmacology, 3D-QSAR, and molecular modeling of (aminoalkyl)benzo- and - thienocycloalkanones as putative atypical antipsychotics
Journal of Medicinal Chemistry, Vol. 42, Núm. 15, pp. 2774-2797
1998
-
Butyrophenone analogues in the carbazole series: Synthesis and determination of affinities at D2 and 5-HT(2A) receptors
Bioorganic and Medicinal Chemistry Letters, Vol. 8, Núm. 24, pp. 3571-3576
1997
-
New cyclic butyrophenone derivatives in the indole series as potential atypical antipsychotics. A simple and practical synthesis of 6-aminomethyl-tetrahydroindol-4-ones and their affinities for D2 and 5-HT(2A) receptors
Bioorganic and Medicinal Chemistry Letters, Vol. 7, Núm. 7, pp. 913-918
1996
-
Synthesis and affinities for dopamine (D2) and 5-hydroxytryptamine (5-HT2A) receptors of 1-(benzoylpropyl)-4-(1-oxocycloalkyl-2-ethyl)-piperazines as cyclic butyrophenone derivatives
Chemical and Pharmaceutical Bulletin, Vol. 44, Núm. 3, pp. 534-541
1995
-
Butyrophenone analogues: Synthesis of 2-methyl-3-ethyl-5-aminoethyl-4,5,6,7-tetrahydroindol-4-ones, and their affinities for d 1 , d 2 and 5-ht 2a receptors
Bioorganic and Medicinal Chemistry Letters, Vol. 5, Núm. 6, pp. 579-584