Publicacións nas que colabora con XERARDO XUSTO GARCIA MERA (42)

2013

  1. Synthesis and allosteric modulation of the dopamine receptor by peptide analogs of l-prolyl-l-leucyl-glycinamide (PLG) modified in the l-proline or l-proline and l-leucine scaffolds

    European Journal of Medicinal Chemistry, Vol. 69, pp. 146-158

2010

  1. Synthesis and pharmacological evaluation of novel 1,3,8- and 1,3,7,8-substituted xanthines as adenosine receptor antagonists

    Bioorganic and Medicinal Chemistry, Vol. 18, Núm. 5, pp. 2001-2009

  2. Synthesis of methyl (±)-3,5-bis(substitutedmethyl)pyrrolidine-2- carboxylates: A convenient approach to proline-mimetics

    Tetrahedron, Vol. 66, Núm. 34, pp. 6797-6805

2009

  1. 1,3-Dialkyl-8-N-substituted benzyloxycarbonylamino-9-deazaxanthines as potent adenosine receptor ligands: Design, synthesis, structure-affinity and structure-selectivity relationships

    Bioorganic and Medicinal Chemistry, Vol. 17, Núm. 10, pp. 3618-3629

  2. Synthesis and biological evaluation of 6-substituted purinylcarbanucleosides with a cyclopenta[b]thiophene pseudosugar

    Synthesis, pp. 2766-2772

  3. Synthesis and pharmacological evaluation of novel 1- and 8-substituted-3-furfuryl xanthines as adenosine receptor antagonists

    Bioorganic and Medicinal Chemistry, Vol. 17, Núm. 18, pp. 6755-6760

2008

  1. Synthesis and antiviral activities of novel purinyl- and pyrimidinyl-carbanucleosides derived from indan

    Synthesis, pp. 1845-1852

  2. Synthesis of novel purinyl-1′-homocarbanucleosides based on a cyclopenta[b]pyrazine system

    Chemical and Pharmaceutical Bulletin, Vol. 56, Núm. 5, pp. 654-658

2007

  1. Probing the anticancer activity of nucleoside analogues: A QSAR model approach using an internally consistent training set

    Journal of Medicinal Chemistry, Vol. 50, Núm. 7, pp. 1537-1545

2006

  1. Synthesis of purinyl and pyrimidinyl 1′(N)-homocarbanucleosides based on a 1-methylcyclopenta[c]pyrazole scaffold; part 2

    Synthesis, pp. 3967-3972

  2. The use of (-)-8-phenylisoneomenthol and (-)-8-phenylmenthol in the enantioselective synthesis of 3-functionalized 2-azabicyclo[2.2.1]heptane derivatives via aza-Diels-Alder reaction

    Tetrahedron, Vol. 62, Núm. 40, pp. 9475-9482

2005

  1. A convenient synthesis of novel pyrimidinyl-5′-nor-1′- homocarbanucleosides based on indanol

    Synthesis, pp. 3549-3554

  2. Enantioselective synthesis of [(1R,3-exo)-2-benzyl-2-azabicyclo[2.2.1]hept- 5-en-3-yl]methanol via Aza-Diels-Alder reaction

    Synlett, pp. 319-321

  3. Experimental and DFT study of the aza-Diels-Alder reaction between cyclopentadiene and protonated benzylimine derivated from glyoxylates

    Tetrahedron, Vol. 61, Núm. 46, pp. 10951-10957

2004

  1. A convenient synthesis of new purinyl-homo-carbonucleosides on a cyclopentane ring fused with pyridazine

    Synthesis, pp. 2855-2862

  2. Anionic ring opening of norbornenes fused to heterocycles

    Tetrahedron, Vol. 60, Núm. 45, pp. 10343-10352

  3. Synthesis of new 6-substituted purinyl-5′-nor-1′- homocarbanucleosides based on indanol

    Tetrahedron, Vol. 60, Núm. 41, pp. 9245-9253

2003

  1. Synthesis and QSAR study of the anticancer activity of some novel indane carbocyclic nucleosides

    Bioorganic and Medicinal Chemistry, Vol. 11, Núm. 23, pp. 4999-5006

  2. The exo-selectivity of the new non-natural chiral auxiliary (+)-(1R,endo)-2-benzonorbornenol in an asymmetric aza-Diels-Alder reaction

    Tetrahedron Letters, Vol. 44, Núm. 3, pp. 431-433

2002

  1. Divergent synthesis of two precursors of 3′-homo-2′-deoxy- and 2′-homo-3′-deoxy-carbocyclic nucleosides

    Tetrahedron, Vol. 58, Núm. 43, pp. 8843-8849