Publikationen in Zusammenarbeit mit Forschern von Universidade Do Porto (14)

2021

  1. Synthesis, Pharmacological, and Biological Evaluation of 2-Furoyl-Based MIF-1 Peptidomimetics and the Development of a General-Purpose Model for Allosteric Modulators (ALLOPTML)

    ACS Chemical Neuroscience, Vol. 12, Núm. 1, pp. 203-215

2016

  1. Novel l-prolyl-l-leucylglycinamide (PLG) tripeptidomimetics based on a 2-azanorbornane scaffold as positive allosteric modulators of the D2R

    Organic and Biomolecular Chemistry, Vol. 14, Núm. 47, pp. 11065-11069

2013

  1. Model for high-throughput screening of multitarget drugs in chemical neurosciences: Synthesis, assay, and theoretic study of rasagiline carbamates

    ACS Chemical Neuroscience, Vol. 4, Núm. 10, pp. 1393-1403

  2. Synthesis and allosteric modulation of the dopamine receptor by peptide analogs of l-prolyl-l-leucyl-glycinamide (PLG) modified in the l-proline or l-proline and l-leucine scaffolds

    European Journal of Medicinal Chemistry, Vol. 69, pp. 146-158

  3. TOPS-MODE model of multiplexing neuroprotective effects of drugs and experimental-theoretic study of new 1,3-rasagiline derivatives potentially useful in neurodegenerative diseases

    Bioorganic and Medicinal Chemistry, Vol. 21, Núm. 7, pp. 1870-1879

2012

  1. A route to selective functionalization of polyhydroxypyrrolidines

    Tetrahedron Letters, Vol. 53, Núm. 9, pp. 1029-1032

2010

  1. Design, synthesis, and evaluation of antineoplastic activity of novel carbocyclic nucleosides

    Molecular Informatics, Vol. 29, Núm. 3, pp. 213-231

  2. Synthesis and pharmacological evaluation of novel 1,3,8- and 1,3,7,8-substituted xanthines as adenosine receptor antagonists

    Bioorganic and Medicinal Chemistry, Vol. 18, Núm. 5, pp. 2001-2009

  3. Synthesis of methyl (±)-3,5-bis(substitutedmethyl)pyrrolidine-2- carboxylates: A convenient approach to proline-mimetics

    Tetrahedron, Vol. 66, Núm. 34, pp. 6797-6805

2009

  1. Synthesis and pharmacological evaluation of novel 1- and 8-substituted-3-furfuryl xanthines as adenosine receptor antagonists

    Bioorganic and Medicinal Chemistry, Vol. 17, Núm. 18, pp. 6755-6760

  2. Synthesis of novel 1-alkyl-8-substituted-3-(3-methoxypropyl) xanthines as putative A2B receptor antagonists

    Bioorganic and Medicinal Chemistry, Vol. 17, Núm. 9, pp. 3426-3432

2008

  1. Synthesis and antiviral activities of novel purinyl- and pyrimidinyl-carbanucleosides derived from indan

    Synthesis, pp. 1845-1852

2006

  1. The use of (-)-8-phenylisoneomenthol and (-)-8-phenylmenthol in the enantioselective synthesis of 3-functionalized 2-azabicyclo[2.2.1]heptane derivatives via aza-Diels-Alder reaction

    Tetrahedron, Vol. 62, Núm. 40, pp. 9475-9482

2004

  1. Synthesis and biological evaluation of carbocyclic nucleosides with 2′,3′-dihomo-xylo-carbocyclic or carbocyclic fused to a tetrahydrofuran ring

    Synthesis, pp. 1991-1995