RUBEN
PRIETO DIAZ
Investigador contratado posdoctoral
Publicaciones (13) Publicaciones de RUBEN PRIETO DIAZ
2024
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Benzylhydroxamic acids as inhibitors of insulin regulated aminopeptidase (IRAP)
European Journal of Medicinal Chemistry Reports, Vol. 12
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Exploring Biginelli-based scaffolds as A2B adenosine receptor antagonists: Unveiling novel structure-activity relationship trends, lead compounds, and potent colorectal anticancer agents
Biomedicine and Pharmacotherapy, Vol. 173
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Progress on the development of Class A GPCR-biased ligands
British Journal of Pharmacology
2023
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Development of Fluorescent 4-[4-(3H-Spiro[isobenzofuran-1,4′-piperidin]-1′-yl)butyl]indolyl Derivatives as High-Affinity Probes to Enable the Study of σ Receptors via Fluorescence-Based Techniques
Journal of Medicinal Chemistry, Vol. 66, Núm. 6, pp. 3798-3817
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Exploring the Effect of Halogenation in a Series of Potent and Selective A2BAdenosine Receptor Antagonists
Journal of Medicinal Chemistry, Vol. 66, Núm. 1, pp. 890-912
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Multicomponent Reaction-Assisted Drug Discovery: A Time- and Cost-Effective Green Approach Speeding Up Identification and Optimization of Anticancer Drugs
International Journal of Molecular Sciences, Vol. 24, Núm. 7
2022
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A 2B adenosine receptor antagonists rescue lymphocyte activity in adenosine-producing patient-derived cancer models
Journal for ImmunoTherapy of Cancer, Vol. 10, Núm. 5
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Exploring Non-orthosteric Interactions with a Series of Potent and Selective A3Antagonists
ACS Medicinal Chemistry Letters, Vol. 13, Núm. 2, pp. 243-249
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Optimization of 2-Amino-4,6-diarylpyrimidine-5-carbonitriles as Potent and Selective A1Antagonists
Journal of Medicinal Chemistry, Vol. 65, Núm. 3, pp. 2091-2106
2021
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3,4-Dihydropyrimidin-2(1H)-ones as Antagonists of the Human A2B Adenosine Receptor: Optimization, Structure-Activity Relationship Studies, and Enantiospecific Recognition
Journal of medicinal chemistry, Vol. 64, Núm. 1, pp. 458-480
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Identification of V6.51L as a selectivity hotspot in stereoselective A2B adenosine receptor antagonist recognition
Scientific Reports, Vol. 11, Núm. 1
2020
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Nitrogen-Walk Approach to Explore Bioisosteric Replacements in a Series of Potent A2B Adenosine Receptor Antagonists
Journal of medicinal chemistry, Vol. 63, Núm. 14, pp. 7721-7739
2017
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Structure-Based Design of Potent and Selective Ligands at the Four Adenosine Receptors
Molecules, Vol. 22, Núm. 11