Publications by the researcher in collaboration with EDDY SOTELO PEREZ (42)

2021

  1. 3,4-Dihydropyrimidin-2(1H)-ones as Antagonists of the Human A2B Adenosine Receptor: Optimization, Structure-Activity Relationship Studies, and Enantiospecific Recognition

    Journal of medicinal chemistry, Vol. 64, Núm. 1, pp. 458-480

2018

  1. Three-Dimensional Printing in Catalysis: Combining 3D Heterogeneous Copper and Palladium Catalysts for Multicatalytic Multicomponent Reactions

    ACS Catalysis, Vol. 8, Núm. 1, pp. 392-404

2017

  1. 3-Oxopyridazin-5-yl-Chalcone Hybrids: Potent Antiplatelet Agents That Prevent Glycoprotein IIb/IIIa Activation

    ChemistrySelect, Vol. 2, Núm. 17, pp. 4920-4933

  2. An efficient and recyclable 3D printed α-Al2O3 catalyst for the multicomponent assembly of bioactive heterocycles

    Applied Catalysis A: General, Vol. 530, pp. 203-210

  3. Enantiospecific Recognition at the A2B Adenosine Receptor by Alkyl 2-Cyanoimino-4-substituted-6-methyl-1,2,3,4-tetrahydropyrimidine-5-carboxylates

    Journal of Medicinal Chemistry, Vol. 60, Núm. 8, pp. 3372-3382

  4. Multicomponent Assembly of the Kinesin Spindle Protein Inhibitor CPUYJ039 and Analogues as Antimitotic Agents

    ACS Combinatorial Science, Vol. 19, Núm. 3, pp. 153-160

2016

  1. 3D printing of a heterogeneous copper-based catalyst

    Journal of Catalysis, Vol. 334, pp. 110-115

2015

  1. Integrated Ugi-Based Assembly of Functionally, Skeletally, and Stereochemically Diverse 1,4-Benzodiazepin-2-ones

    Journal of Organic Chemistry, Vol. 80, Núm. 3, pp. 1533-1549

  2. Pyrazin-2(1H)-ones as a novel class of selective A3 adenosine receptor antagonists

    Future Medicinal Chemistry, Vol. 7, Núm. 11, pp. 1373-1380

  3. Sol-gel entrapped Cu in a silica matrix: An efficient heterogeneous nanocatalyst for Huisgen and Ullmann intramolecular coupling reactions

    Applied Catalysis A: General, Vol. 502, pp. 86-95

2014

  1. Structure-based design of new KSP-Eg5 inhibitors assisted by a targeted multicomponent reaction

    ChemBioChem, Vol. 15, Núm. 10, pp. 1471-1480

2013

  1. Copper-catalyzed huisgen 1,3-dipolar cycloaddition under oxidative conditions: Polymer-assisted assembly of 4-acyl-1-substituted-1,2,3-triazoles

    Journal of Organic Chemistry, Vol. 78, Núm. 13, pp. 6540-6549

  2. Discovery of 3,4-dihydropyrimidin-2(1 H)-ones as a novel class of potent and selective A2B adenosine receptor antagonists

    ACS Medicinal Chemistry Letters, Vol. 4, Núm. 11, pp. 1031-1036

  3. Multicomponent assembly of diverse pyrazin-2(1 H)-one chemotypes

    Journal of Organic Chemistry, Vol. 78, Núm. 9, pp. 4402-4409

  4. Selective and potent adenosine A3 receptor antagonists by methoxyaryl substitution on the N-(2,6-diarylpyrimidin-4-yl)acetamide scaffold

    European Journal of Medicinal Chemistry, Vol. 59, pp. 235-242

  5. Three-component assembly of structurally diverse 2-aminopyrimidine-5- carbonitriles

    ACS Combinatorial Science, Vol. 15, Núm. 7, pp. 370-378

2012

  1. Discovery and preliminary SAR of 5-arylidene-2,2-dimethyl-1,3-dioxane-4,6- diones as platelet aggregation inhibitors

    Combinatorial Chemistry and High Throughput Screening, Vol. 15, Núm. 7, pp. 551-554

2011

  1. Convergent assembly of structurally diverse quinazolines

    Organic and Biomolecular Chemistry, Vol. 9, Núm. 2, pp. 351-357

  2. Pyrimidine derivatives as potent and selective A3 adenosine receptor antagonists

    Journal of Medicinal Chemistry, Vol. 54, Núm. 2, pp. 457-471

  3. Silica-supported aluminum chloride-assisted solution phase synthesis of pyridazinone-based antiplatelet agents

    ACS Combinatorial Science, Vol. 13, Núm. 1, pp. 7-12