Publications by the researcher in collaboration with Luis Castedo Expósito (118)

2012

  1. Synthesis of 3-alkyl enol mimics inhibitors of type II dehydroquinase: Factors influencing their inhibition potency

    Organic and Biomolecular Chemistry, Vol. 10, Núm. 18, pp. 3662-3676

2011

  1. A prodrug approach for improving antituberculosis activity of potent mycobacterium tuberculosis type II dehydroquinase inhibitors

    Journal of Medicinal Chemistry, Vol. 54, Núm. 17, pp. 6063-6084

  2. Benzenediazonium-2-carboxylate

    Encyclopedia of Reagents for Organic Synthesis

  3. Six-Membered Heterocycles: Pyridines

    Modern Heterocyclic Chemistry (Wiley-VCH), pp. 1431-1525

  4. Tetrahydrobenzothiophene Derivatives: Conformationally Restricted Inhibitors of TypeII Dehydroquinase

    ChemMedChem, Vol. 6, Núm. 2, pp. 266-272

2010

  1. Synthesis and biological evaluation of new nanomolar competitive inhibitors of Helicobacter pylori type II dehydroquinase. Structural details of the role of the aromatic moieties with essential residues

    Journal of Medicinal Chemistry, Vol. 53, Núm. 1, pp. 191-200

  2. Understanding the key factors that control the inhibition of type II dehydroquinase by (2R)-2-benzyl-3-dehydroquinic acids

    ChemMedChem, Vol. 5, Núm. 10, pp. 1726-1733

2009

  1. 2-Substituted-3-dehydroquinic acids as potent competitive inhibitors of type II dehydroquinase

    ChemMedChem, Vol. 4, Núm. 12, pp. 1980-1984

  2. A selective resin for trans-diequatorial-1,2-diols

    Tetrahedron Letters, Vol. 50, Núm. 16, pp. 1795-1798

2008

  1. Competitive inhibitors of Helicobacter pylori type II dehydroquinase: Synthesis, biological evaluation, and NMR studies

    ChemMedChem, Vol. 3, Núm. 5, pp. 756-770

  2. Stereoselective synthesis of novel cyclic γ-amino acids and triazole derivatives

    European Journal of Organic Chemistry, pp. 3991-4003

  3. The conformational rigidity of butane-1,2-diacetals as a powerful synthetic tool

    Chemical Society Reviews, Vol. 37, Núm. 8, pp. 1689-1708

2007

  1. Nanomolar competitive inhibitors of Mycobacterium tuberculosis and Streptomyces coelicolor type II dehydroquinase

    ChemMedChem, Vol. 2, Núm. 2, pp. 194-207

  2. Product Class 5: Phenols and Phenolates

    Science of Synthesis: Houben-Weyl Methods of Molecular Transformations Vol. 31a

  3. Progress in type II dehydroquinase inhibitors: From concept to practice

    Medicinal Research Reviews, Vol. 27, Núm. 2, pp. 177-208

  4. Synthesis by Elimination

    Science of Synthesis: Houben-Weyl Methods of Molecular Transformations Vol. 31a

  5. Synthesis by Rearrangement

    Science of Synthesis: Houben-Weyl Methods of Molecular Transformations Vol. 31a

  6. Synthesis with Retention of the Functional Group

    Science of Synthesis: Houben-Weyl Methods of Molecular Transformations Vol. 31a

2006

  1. Determination of the bound conformation of a competitive nanomolar inhibitor of Mycobacterium tuberculosis type II dehydroquinase by NMR spectroscopy

    ChemMedChem, Vol. 1, Núm. 9, pp. 990-996

  2. Synthesis and reactivity of new strained cyclic allene and alkyne precursors

    Pure and Applied Chemistry